中文名 | Ca2+ channel agonist 1 |
英文名 | Ca2+ channel agonist 1 |
别名 | 化合物CA2+ CHANNEL AGONIST 1 CDK2抑制剂(CA2+ CHANNEL AGONIST 1) |
英文别名 | Ca2+ channel agonist 1 1-Butanol, 2-[[6-[(phenylmethyl)amino]-9-propyl-9H-purin-2-yl]amino]-, (2R)- |
CAS | 1402821-24-2 |
化学式 | C19H26N6O |
分子量 | 354.45 |
溶解度 | 10毫米DMSO |
存储条件 | -20℃ |
体外研究 | Ca 2+ channel agonist 1 (Compound 13d) is an agonist of N-type Ca 2+ channel and an inhibitor of Cdk2, with EC 50 s of 14.23 μM and 3.34 μM, respectively. Ca 2+ channel agonist 1 exhibits a ca. 2-fold increased agonism and a 22-fold decreased cdk2 kinase activity versus the standard, (R)-roscovitine. |
1mg | 5mg | 10mg | |
---|---|---|---|
1 mM | 2.821 ml | 14.106 ml | 28.213 ml |
5 mM | 0.564 ml | 2.821 ml | 5.643 ml |
10 mM | 0.282 ml | 1.411 ml | 2.821 ml |
5 mM | 0.056 ml | 0.282 ml | 0.564 ml |
微信搜索化工百科或扫描下方二维码,添加化工百科小程序,随时随地查信息!